Sodium ya Closantel

Ibisobanuro bigufi:

Umubare wa CAS :61438-64-0

Inzira ya molekulari:C23H15Cl2I2N2NaO4


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Sodium ya Closantel

Sodium ya Closantel ni anthelmintic yagutse, igira ingaruka nziza kuri trematode zitandukanye, nematode na arthropod larvae;ibikorwa byayo birwanya fluke birwanya cyane cyane Fasciola hepatica, anti-nematode hamwe nigikorwa cyo kurwanya indwara ya arthropodes igamije ahanini inyo zose zonsa amaraso cyangwa plasma.
Iki gicuruzwa gikoreshwa cyane mu kwandura indwara zanduye zavuzwe haruguru mu nka n'intama.Irashobora gutangwa mu kanwa cyangwa kubabyeyi (munsi yubutaka no mumitsi), kandi ifite ingaruka zo kuvura no gukumira.Hano hari inshinge, ibinini hamwe nogukoresha isoko.Mubisanzwe, irahujwe na mebendazole nibindi bicuruzwa bya benzimidazole kugirango ikore intungamubiri yintama;irahujwe na levamisole gukora ibinini bigizwe ninka.

Closantel-Sodium- (1)

Uburyo bwibikorwa nibiranga

Sodium ya Closalamide izwi kandi nka chlorsalamide umunyu wa sodium n'umunyu wa chlorsalamide.Ni mubice bimwe bya salicylanilide hamwe na iodosalamide kandi ni ubwoko bushya bwa anti-parasitike yagutse ikoreshwa mubworozi.Ubuvuzi bw’udukoko, isura ni ifu yumuhondo gake, idafite impumuro nziza cyangwa impumuro nkeya, gushonga byoroshye muri Ethanol cyangwa acetone, gushonga muri methanol, no kudashonga mumazi cyangwa chloroform.Igikorwa cya farumasi nuguhagarika inzira ya fosifora ya mitochondial yinyo, bityo bikarinda synthesis ya adenosine triphosphate (ATP) yinyo, biganisha ku kugabanuka kwihuse kwingufu za metabolisme yinyo hanyuma amaherezo apfa.Sodium ya Closantel irashobora kwica burundu ibisebe, ibisebe byamaraso, inzoka zinzoka, strongyloide, impyiko nematode, ibiboko, burrow nematode, supine umunwa nematode, imirasire esophagus Flukes, capillary nematode, isazi yuruhu, intama izunguruka isazi, amatiku, ibisebe, ibisebe, nematode, Fasciola hepatica, isazi yo mu gifu isazi, lipoma canis nizindi nkoko zo mu bwoko bwimbere ninyuma.Ifite ingaruka nziza kuri livre ya trematode zitandukanye, nematode na arthropods;ibikorwa byayo byo kurwanya anti-fluke ahanini ni ibya Fasciola hepatica, kandi ibikorwa byayo byo kurwanya nematode na arthropods bigenewe cyane cyane ibinyobwa bitandukanye.Umubiri winyo wamaraso cyangwa plasma.Ibizamini bya Clinical efficacy byerekanye ko iyo bikozwe ku gipimo cya 10 mg / kg cy'umubiri, bigira ingaruka zuzuye ku ntama Fasciola hepatica, imbere na inyuma ya disiki ya trematode, ibihaha hamwe na nematode nyinshi zo mu gifu no mu mubiri.Ningaruka nziza yo kwangiza intama.Igipimo cyiza.

Imyiteguro

5%, 10% inshinge ya sodium ya Closantel;
1% Ivermectin + 12,5% inshinge ya sodium ya Closantel;
5%, 10% Guhagarika sodium ya Closantel.


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